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ECTRIMS 2025

Cree B, et al. Long-Term Efficacy and Safety of Ublituximab in Relapsing Multiple Sclerosis: Results from 6 Years of ULTIMATE I and II Open-Label Extension (ECTRIMS 9.24.25)

Hersh C, et al. Real world clinical experience from ENABLE, the first Phase 4 observational study for patients with relapsing multiple sclerosis initiating ublituximab (ECTRIMS 9.24.25)

Singer B, et al. Safety and Tolerability of a Modified Ublituximab Dosing Regimen: Updates from the ENHANCE Study (ECTRIMS 9.24.25)

CMSC 2025

Cree B, et al. No association between decreases in serum immunoglobulin (Ig) levels below lower limit of normal (LLN) and serious infections (SI) with long term ublituximab (UBL) treatment in patients with Relapsing Multiple Sclerosis (RMS) (CMSC 5.29.25)

Fox E, et al. Retrospective Evaluation of Infusion Tolerability: Ublituximab Real-World Observational Survey (ENAMOR) (CMSC 5.29.25)

Foley J, et al. Safety and Tolerability of 30-minute Ublituximab Infusions: Updates from the ENHANCE Study (CMSC 5.29.25)

AAN 2025

Cree B, et al. Five Years of Ublituximab in Relapsing Multiple Sclerosis: Results from the Open- Label Extension of ULTIMATE I and II Studies (AAN 4.9.25)

Foley J, et al. Safety and Tolerability of a Modified Dosing Regimen of Ublituximab: Updates from the ENHANCE Study (AAN 4.9.25)

Fox E, et al. Retrospective Evaluation of Infusion Tolerability: Ublituximab Real-World Observational Survey (ENAMOR) (AAN 4.7.25)

Fox, E, et al. ENABLE: the first phase 4 observational study for patients with relapsing MS treated with ublituximab in real world clinical settings (AAN 4.7.25)

Steinman L, et al. No association between decreases in serum immunoglobulin (Ig) levels below lower limit of normal (LLN) and serious infections (SI) with long-term ublituximab (UBL) treatment in patients with relapsing Multiple Sclerosis (RMS) (AAN 4.7.25)

ACTRIMS 2025

Foley J, et al. Safety and Tolerability of 30-minute Ublituximab Infusions: Updates from the ENHANCE Study (ACTRIMS 2.27.25)

Monson N, et al. The Design of a Study to Evaluate Fc Biology and Genetic Diversity in Multiple Sclerosis (ACTRIMS 2.27.25)

OUR PUBLICATION LIBRARY

We welcome you to explore our comprehensive publications database. All publications are available to download. Please select one or more fields from the list below to help narrow your search.
DateTitleAuthorDrugConferencesFilehf:tax:month-yearhf:tax:conferencehf:tax:therapeuticshf:tax:drug
09/24/2025Safety and Tolerability of a Modified Ublituximab Dosing Regimen: Updates from the ENHANCE Studyet al., Singer Bublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2025european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
09/24/2025Real world clinical experience from ENABLE, the first Phase 4 observational study for patients with relapsing multiple sclerosis initiating ublituximabet al., Hersh Cublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2025european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
09/24/2025Long-Term Efficacy and Safety of Ublituximab in Relapsing Multiple Sclerosis: Results from 6 Years of ULTIMATE I and II Open-LabelCree B, et al.ublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2025european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
05/29/2025Safety and Tolerability of 30-minute Ublituximab Infusions: Updates from the ENHANCE Studyet al., Foley Jublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2025annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
05/29/2025Retrospective Evaluation of Infusion Tolerability: Ublituximab Real-World Observational Survey (ENAMOR)et al., Fox Eublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2025annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
05/29/2025No association between decreases in serum immunoglobulin (Ig) levels below lower limit of normal (LLN) and serious infections (SI) with long term ublituximab (UBL) treatment in patients with Relapsing Multiple Sclerosis (RMS)Cree B, et al.ublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2025annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
04/09/2025Five Years of Ublituximab in Relapsing Multiple Sclerosis: Results from the OpenLabel Extension of ULTIMATE I and II StudiesCree B, et al.ublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2025american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/09/2025Safety and Tolerability of a Modified Dosing Regimen of Ublituximab: Updates from the ENHANCE Studyet al., Foley Jublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2025american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/07/2025No association between decreases in serum immunoglobulin (Ig) levels below lower limit of normal (LLN) and serious infections (SI) with long-term ublituximab (UBL) treatment in patients with relapsing Multiple Sclerosis (RMS)et al., Steinman Lublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2025american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/07/2025ENABLE: the first phase 4 observational study for patients with relapsing MS treated with ublituximab in real world clinical settingset al., Fox Eublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2025american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/07/2025Retrospective Evaluation of Infusion Tolerability: Ublituximab Real-World Observational Survey (ENAMOR)et al., Fox Eublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2025american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/03/2025Switching to ublituximab from prior anti-CD20 monoclonal antibody therapy: a case report seriesBerkovich R, et al.ublituximab (TG-1101)Frontiers in Neurology Journal2025frontiers-in-neurology-journalautoimmuneublituximab-tg-1101
04/03/2025The Evolution of Anti-CD20 Treatment for Multiple Sclerosis: Optimization of Antibody Characteristics and FunctionCree B, et al.ublituximab (TG-1101)CNS Drugs2025cns-drugsautoimmuneublituximab-tg-1101
02/27/2025Safety and Tolerability of 30-minute Ublituximab Infusions: Updates from the ENHANCE Studyet al., Foley Jublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2025americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
02/27/2025The Design of a Study to Evaluate Fc Biology and Genetic Diversity in Multiple Sclerosiset al., Monson Nublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2025americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
10/23/2024Improvements in no evidence of disease activity with ublituximab vs. teriflunomide in the ULTIMATE phase 3 studies in relapsing multiple sclerosisAlvarez E, et al.ublituximab (TG-1101)Frontiers in Neurology Journal2024frontiers-in-neurology-journalautoimmuneublituximab-tg-1101
09/18/2024Comparison of Multiple Sclerosis Disease Activity (MSDA) Test Results Between Patients Treated with Ublituximab and Teriflunomide in the Phase 3 ULTIMATE I and II Studieset al., Foley Jublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2024european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
09/18/2024Five Years of Ublituximab in Relapsing Multiple Sclerosis: Results from the Open-Label Extension of ULTIMATE I and II StudiesCree B, et al.ublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2024european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
09/18/2024Efficacy and Tolerability of Ublituximab after Transitioning from a Different Disease-Modifying Therapy: Updates from the ENHANCE Studyet al., Foley Jublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2024european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
05/30/2024BRIUMVI® Pregnancy Registry: A Prospective Study of Pregnancy and Infant Outcomes in Patients Treated with BRIUMVI (ublituximab-xiiy)Bove R, et al.ublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2024annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
05/30/2024A Post-Marketing Study Evaluating the Presence and Concentration of BRIUMVI®(ublituximab-xiiy) in Breastmilk (PROVIDE)Bove R, et al.ublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2024annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
04/17/2024Early Initiation of Ublituximab Treatment is Associated with Improved Disability Outcomes Among Treatment-Naïve Participants in ULTIMATE I and IIet al., Robertson Dublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2024american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/17/2024Ublituximab Significantly Reduces Radiological Disease Activity at 12 Weeks: Post-hoc analysis of Participants with Highly Active Disease in the ULTIMATE I & II Phase 3 Studieset al., Robertson Dublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2024american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/14/2024MS Relapse Redefined: Distinguishing True Relapses from Pseudoexacerbations in the ULTIMATE I and II Trials Comparing Ublituximab vs Teriflunomideet al., Krieger Sublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2024american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
02/29/2024Evaluating the Maintenance of Efficacy and Tolerability of Transitioning from IV Anti-CD20 Therapy to Ublituximab: ENHANCE Study Interim Dataet al., Singer Bublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2024americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
02/29/2024MS Relapse Redefined: Addressing the Radiological/Pseudoexacerbation Paradox with High Efficacy Therapy in the ULTIMATE I and II TrialsAlvarez E, et al.ublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2024americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
10/12/2023Disease Activity Score and Disease Pathway Scores Measured Using the Multiple Sclerosis Disease Activity Test are Significantly Reduced Prior to the Week 96 Dose for Patients Treated with Ublituximab in the Phase 3 ULTIMATE I and II Studieset al., Foley Jublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2023european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/11/2023Evaluating the Maintenance of Efficacy and Tolerability when Transitioning from IV anti-CD20 Therapy to Ublituximab: ENHANCE Study Design, Patient Demographics and Preliminary Dataet al., Foley Jublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2023european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/11/2023Ublituximab Reduces Thalamic Volume Loss and New Lesion Formation in Participants of the ULTIMATE I & II Phase 3 StudiesArnold D, et al.ublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2023european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
06/01/2023Ublituximab Is Associated with Significant Improvement in Fatigue: Results from Ultimate I and IIAlvarez E, et al.ublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2023annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
04/25/2023Ublituximab, a Novel, Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), Demonstrates Enhanced Antibody-Dependent Cellular Cytolysis (ADCC) Relative to Other Anti-CD20 mAbset al., Foley Jublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2023american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/24/2023Ublituximab Efficacy in Treatment-Naive Participants With Relapsing Multiple Sclerosis in the Phase 3 ULTIMATE I and II Studieset al., Steinman Lublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2023american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/24/2023Disease Outcomes With Ublituximab in Participants With Highly Active Disease: Subpopulation Analyses of the Phase 3 ULTIMATE I and II Studies in Participants With Relapsing Multiple SclerosisAlvarez E, et al.ublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2023american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
02/23/2023Onset and Maintenance of No Evidence of Disease Activity With Ublituximab: Analyses of the Phase 3 ULTIMATE I and II Studies in Participants With Relapsing Multiple SclerosisAlvarez E, et al.ublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2023americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
02/23/2023Early, Transient Shift in Hematologic Parameters Observed With Ublituximab in the ULTIMATE I and II Phase 3 Studieset al., Qian Publituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2023americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
12/11/2022First-in-Human (FIH) Study of the Fully-Human Kappa-Lambda CD19/CD47 Bispecific Antibody TG-1801 in Patients (pts) with BCell LymphomaChea C, et al.TG-1801American Society of Hematology Annual Meeting (ASH)2022american-society-of-hematology-annual-meeting-ashoncologytg-1801
10/26/2022Functional Systems Scores and Expanded Disability Status Scale Score Evaluations in the ULTIMATE I and II Studies of Ublituximab Versus Teriflunomide in Participants With Relapsing Multiple SclerosisCree B, et al.ublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2022european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/26/2022Disability Changes in the Absence of Relapse in the Phase 3 ULTIMATE I and II Studies of Ublituximab Versus Teriflunomide in Participants With Relapsing Multiple Sclerosiset al., Wray Sibylublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2022european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/26/2022Ublituximab Treatment Is Associated With a Significant Proportion of Participants Achieving NEDA-4Alvarez E, et al.ublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2022european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/26/2022Disease Outcomes With Ublituximab in Treatment-Naive Participants: Subpopulation Analyses of the Phase 3 ULTIMATE I and II Studies in Participants With Relapsing Multiple Sclerosiset al., Steinman Lublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2022european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/26/2022B-Cell Depletion and Return in Participant Subgroups of the Phase 3 ULTIMATE I and II Studies of Ublituximab Versus Teriflunomide in Participants With Relapsing Multiple Sclerosiset al., Fox Eublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2022european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
08/25/2022Ublituximab versus Teriflunomide in Relapsing Multiple Sclerosiset al., Steinman Lublituximab (TG-1101)New England Journal of Medicine (NEJM)2022new-england-journal-of-medicine-nejmautoimmuneublituximab-tg-1101
06/27/2022Improved Quality of Life With Ublituximab in the ULTIMATE I and II Studies in Relapsing Multiple Sclerosiset al., Selmaj Kublituximab (TG-1101)5th Congress of the European Academy of Neurology (EAN)20225th-congress-of-the-european-academy-of-neurology-eanautoimmuneublituximab-tg-1101
06/27/2022Disability Improvements With Ublituximab in Relapsing Multiple Sclerosis: Pooled Post Hoc Analyses of the ULTIMATE I and II StudiesCree B, et al.ublituximab (TG-1101)5th Congress of the European Academy of Neurology (EAN)20225th-congress-of-the-european-academy-of-neurology-eanautoimmuneublituximab-tg-1101
06/26/2022Ublituximab Efficacy Outcomes in Relapsing Multiple Sclerosis Patient Subgroups in the ULTIMATE I and II Studieset al., Hartung Publituximab (TG-1101)5th Congress of the European Academy of Neurology (EAN)20225th-congress-of-the-european-academy-of-neurology-eanautoimmuneublituximab-tg-1101
06/02/2022Improved Cognitive Processing Speed With Ublituximab in Patients With Highly Active Relapsing Multiple Sclerosiset al., Robertson Dublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2022annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
06/02/2022Infusion-Related Reactions With Ublituximab in the Phase 3 ULTIMATE I and II Studies in Relapsing Multiple Sclerosiset al., Fox Eublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2022annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
06/02/2022Reduced Disease Progression With Ublituximab vs Teriflunomide in the Phase 3 ULTIMATE I and II Studies in Relapsing Multiple SclerosisAlvarez E, et al.ublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2022annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
04/05/2022Relapse Rate and Time to First Relapse were Improved with Ublituximab vs Teriflunomide in the Phase 3 ULTIMATE I and ULTIMATE II Studies in Patients with Relapsing Multiple Sclerosis (RMS)et al., Steinman Lublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2022american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/03/2022Disability Improvements with Ublituximab in Relapsing Multiple Sclerosis (RMS): Expanded Disability Status Scale (EDSS), 9-Hole Peg Test (9-HPT), and Timed 25-Foot Walk (T25FW) Evaluations from the Phase 3 ULTIMATE I and II StudiesCree B, et al.ublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2022american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/03/2022Ublituximab Treatment is Associated with a Significant Proportion of Patients Achieving No Evidence of Disease Activity (NEDA): Results from the Ultimate I and Ultimate II Phase 3 Studies of Ublituximab vs Teriflunomide in Relapsing Multiple Sclerosis (RMS)Alvarez E, et al.ublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2022american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/03/2022Infusion-Related Reactions (IRRs) with Ublituximab in Patients with Relapsing Multiple Sclerosis (RMS): Post Hoc Analyses from the Phase 3 ULTIMATE I and II Studieset al., Fox Eublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2022american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
02/24/2022Reduction in T1 Hypointense Lesions with Ublituximab vs Teriflunomide in the Phase 3 ULTIMATE I & II Studies in Relapsing Multiple SclerosisCree B, et al.ublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2022americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
02/24/2022Pharmacodynamics of B-Cell Depletion and Pharmacokinetics of the Novel Anti-CD20 Monoclonal Antibody Ublituximab in Patients with Relapsing Multiple Sclerosiset al., Fox Eublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2022americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
02/24/2022Neutralizing Antibodies and Antidrug Antibodies in the Ublituximab Phase 3 ULTIMATE I & II Studies in Relapsing Multiple SclerosisAlvarez E, et al.ublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2022americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
12/13/2021Favorable Outcomes for Patients with Co-morbidities or Concomitant Medications Treated with U2: A Retrospective Analysis of UNITY-CLL Phase 3 Trialet al., Pinilla-Ibarz Jublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2021american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/13/2021Efficacy and Safety of Ublituximab in Combination with Umbralisib (U2) in Patients with Chronic Lymphocytic Leukemia (CLL) by Treatment Status: A Sub-analysis of the Phase 3 UNITY-CLL Studyet al., Jacobs RAmerican Society of Hematology Annual Meeting (ASH)2021american-society-of-hematology-annual-meeting-ashoncology
12/12/2021A Phase 2 Study Evaluating the Addition of Ublituximab and Umbralisib (U2) to Ibrutinib in Patients with Chronic Lymphocytic Leukemia (CLL): a Minimal Residual Disease (MRD)-driven, Time-limited Approachet al., Roeker Lublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2021american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/12/2021Efficacy and Safety of Umbralisib and Ublituximab (U2), and U2 Plus Bendamustine in Patients with Relapsed or Refractory Diffuse Large B-cell Lymphoma (DLBCL)Burke J, et al.ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2021american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/11/2021The Combination of Umbralisib Plus Ublituximab is Active in Patients with Relapsed or Refractory Marginal Zone Lymphoma (MZL): Results from the Phase 2 Global UNITY-NHL TrialChavez J, et al.ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2021american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/11/2021The Selective Bruton’s Tyrosine Kinase (BTK) Inhibitor TG-1701 as Monotherapy and in Combination with Ublituximab and Umbralisib (U2) in Patients with B-cell MalignanciesCheah C, et al.ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2021american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
10/14/2021Ublituximab Is Associated With Significant Improvement in the Multiple Sclerosis Functional Composite (MSFC): Results From the Phase 3 ULTIMATE I & II Studieset al., Steinman Lublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2021european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/14/2021Phase 3 Results of the ULTIMATE I & II Global Studies: Ublituximab Versus Teriflunomide in Relapsing Multiple Sclerosiset al., Steinman Lublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2021european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
09/21/2021Integrated Safety Analysis of Umbralisib, a Dual PI3Kδ/CK1ε Inhibitor, in Relapsed/Refractory Lymphoid MalignanciesDavids M, et al.umbralisib (TGR-1202)Blood Advances Journal – published by The American Society of Hematology2021blood-advances-journal-published-by-the-american-society-of-hematologyoncologyumbralisib-tgr-1202
09/19/2021A Phase 1/2 Study of Umbralisib, Ublituximab, and Venetoclax in Patients with Relapsed or Refractory Chronic Lymphocytic Leukemia (CLL)Barr, P et al.TG-1701, ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2021international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologytg-1701 ublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
09/19/2021TG-1701, a Selective Bruton Tyrosine Kinase (BTK) Inhibitor, as Monotherapy and in Combination with Ublituximab and Umbralisib (U2) in Patients with Chronic Lymphocytic LeukemiaCheah C, et al.International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2021international-workshop-on-chronic-lymphocytic-leukemia-iwclloncology
09/18/2021Phase I/II Study of Umbralisib (TGR-1202), Ublituximab (TG-1101), and Pembrolizumab in Patients with Relapsed or Refractory Chronic Lymphocytic Leukemia and Richter’s Transformation: 5-Year Follow-upet al., Roeker Lublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2021international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
09/18/2021Umbralisib Plus Ublituximab (U2) Is Superior to Obinutuzumab Plus Chlorambucil (O+Chl) in Patients with Treatment-Naïve (TN) and Relapsed/Refractory (R/R) Chronic Lymphocytic Leukemia (CLL): Results from the Phase 3 UNITY-CLL Studyet al., Jurczak Wublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2021international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
09/18/2021Phase I/II Study of Umbralisib (TGR-1202), Ublituximab (TG-1101), and Pembrolizumab in Patients with Relapsed or Refractory Chronic Lymphocytic Leukemia and Richter’s Transformation: 5-Year Follow-upet al., Roeker Lublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
06/18/2021Antitumoral Activity of the Novel BTK Inhibitor TG-1701 is Associated with Disruption of Ikaros Signaling and Improvement of Anti-CD20 Therapy in B-cell Non-Hodgkin Lymphomaet al., Roue GTG-1701International Congress on Malignant Lymphoma (ICML)2021international-congress-on-malignant-lymphoma-icmloncologytg-1701
06/18/2021Updated Results of the Selective Bruton Tyrosine kinase (BTK) Inhibitor TG-1701, as Monotherapy and in Combination with Ublituximab and Umbralisib (U2) in Patients (pts) with B-cell MalignanciesCheah C, et al.TG-1701, ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)International Congress on Malignant Lymphoma (ICML)2021international-congress-on-malignant-lymphoma-icmloncologytg-1701 ublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
06/18/2021Ublituximab versus Teriflunomide in Relapsing Multiple Sclerosis: Results of the Phase 3 ULTIMATE I and II Trialset al., Steinman Lublituximab (TG-1101)5th Congress of the European Academy of Neurology (EAN)20215th-congress-of-the-european-academy-of-neurology-eanautoimmuneublituximab-tg-1101
06/11/2021Updated Results of the Selective Bruton Tyrosine Kinase (BTK) Inhibitor TG-1701, as Monotherapy and in Combination with Ublituximab and Umbralisib (U2) in Patients (pts) with B-cell MalignanciesCheah C, et al.Congress of the European Hematology Association (EHA)2021congress-of-the-european-hematology-association-ehaoncology
06/04/2021Updated Results of the Selective Bruton Tyrosine Kinase (BTK) Inhibitor TG-1701, as Monotherapy and in Combination with Ublituximab and Umbralisib(U2) in Patients (pts) with B-cell MalignanciesCheah C, et al.TG-1701, ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Clinical Oncology Annual Meeting (ASCO)2021american-society-of-clinical-oncology-annual-meeting-ascooncologytg-1701 ublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
06/04/2021VIDEO: Updated Results of the Selective Bruton Tyrosine Kinase (BTK) Inhibitor TG-1701, as Monotherapy and in Combination with Ublituximab and Umbralisib (U2) in Patients (pts) with B-cell MalignanciesCheah C, et al.TG-1701, ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Clinical Oncology Annual Meeting (ASCO)2021american-society-of-clinical-oncology-annual-meeting-ascooncologytg-1701 ublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
04/17/2021Efficacy and Safety of Ublituximab vs Teriflunomide in Patients with Relapsing Multiple Sclerosis: Results from Two Phase 3 Studies ULTIMATE I & ULTIMATE II American Academy of Neurologyet al., Steinman Lublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2021american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
03/09/2021Umbralisib, a Dual PI3Kδ/CK1ε Inhibitor in Patients with Relapsed/Refractory Indolent Lymphomaet al., Fowler Numbralisib (TGR-1202)Journal of Clinical Oncology2021journal-of-clinical-oncologyoncologyumbralisib-tgr-1202
02/22/2021A Phase 3, Randomized Trial of Ublituximab Plus Ibrutinib for Patients with Relapsed/Refractory High-Risk Chronic Lymphocytic Leukaemiaet al., Sharman Jublituximab (TG-1101)THE LANCET Haematology2021the-lancet-haematologyublituximab-tg-1101
12/07/2020A Phase 1/2 Study of Umbralisib Ublituximab and Venetoclax in Patients with Relapsed or Refractory Chronic Lymphocytic Leukemia (CLL)Barr P, et al.ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/07/2020Umbralisib, a PI3Kδ/CK1ε dual inhibitor demonstrates marked clinical activity in patients with relapsed or refractory indolent non-Hodgkin lymphoma: Results from the Phase 2 global UNITY-NHL trialet al., Zinzani Pumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/07/2020Phase 3 Study of Umbralisib Combined With Ublituximab vs Obinutuzumab Plus Chlorambucil in Patients With Chronic Lymphocytic Leukemia: Results From UNITY-CLLet al., Gribben Jublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/07/2020VIDEO: Phase 3 Study of Umbralisib Combined With Ublituximab vs Obinutuzumab Plus Chlorambucil in Patients With Chronic Lymphocytic Leukemia: Results From UNITY-CLLGribben, J et al.ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/07/2020VIDEO: Umbralisib, a PI3Kδ/CK1ε dual inhibitor demonstrates marked clinical activity in patients with relapsed or refractory indolent non-Hodgkin lymphoma: Results from the Phase 2 global UNITY-NHL trialP et al., Zinzaniumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/07/2020VIDEO: A Phase 1/2 Study of Umbralisib Ublituximab and Venetoclax in Patients with Relapsed or Refractory Chronic Lymphocytic Leukemia (CLL)Barr, P et al.ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/05/2020Clinical Activity of TG-1701, As Monotherapy and in Combination with Ublituximab and Umbralisib (U2), in Patients with B-Cell MalignanciesCheah C, et al.TG-1701, ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologytg-1701 ublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/05/2020VIDEO: Clinical Activity of TG-1701, As Monotherapy and in Combination with Ublituximab and Umbralisib (U2), in Patients with B-Cell MalignanciesCheah C, et al.TG-1701, ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologytg-1701 ublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
12/02/2020Phase 2 Study of the Safety and Efficacy of Umbralisib in Patients with CLL Who Are Intolerant to BTK or PI3Kδ Inhibitor Therapyet al., Mato Aumbralisib (TGR-1202)Blood Medical Journal – published by the American Society of Hematology (Blood)2020blood-medical-journal-published-by-the-american-society-of-hematology-bloodoncologyumbralisib-tgr-1202
11/04/2020Umbralisib Plus Ublituximab (U2) Is Superior to Obinutuzumab Plus Chlorambucil (O+Chl) in Patients with Treatment Naïve (TN) and Relapsed/Refractory (R/R) Chronic Lymphocytic Leukemia (CLL): Results from the Phase 3 UNITY-CLL Studyet al., Gribben Jublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
11/04/2020Umbralisib, the Once Daily Dual Inhibitor of PI3Kδ and Casein Kinase-1ε Demonstrates Clinical Activity in Patients with Relapsed or Refractory Indolent Non-Hodgkin Lymphoma: Results from the Phase 2 Global UNITY-NHL Trialet al., Zinzani Pumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
11/04/2020A Phase 1/2 Study of Umbralisib, Ublituximab, and Venetoclax (U2-Ven) in Patients with Relapsed or Refractory Chronic Lymphocytic Leukemia (CLL)Barr P, et al.ublituximab (TG-1101), umbralisib (TGR-1202), umbralisib + ublituximab (U2)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202 umbralisib-ublituximab-u2
11/04/2020Clinical Activity of TG-1701, As Monotherapy and in Combination with Ublituximab and Umbralisib (U2), in Patients with B-Cell MalignanciesCheah C, et al.TG-1701, ublituximab (TG-1101), umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2020american-society-of-hematology-annual-meeting-ashoncologytg-1701 ublituximab-tg-1101 umbralisib-tgr-1202
07/08/2020The Dual PI3Kδ/CK1ε Inhibitor Umbralisib Exhibits Unique Immunomodulatory Effects on CLL T CellsPinilla-Ibarz J. et al.umbralisib (TGR-1202)Blood Advances Journal – published by The American Society of Hematology2020blood-advances-journal-published-by-the-american-society-of-hematologyoncologyumbralisib-tgr-1202
06/22/2020TG-1701, a Novel Irreversible Bruton’s Kinase (BTK) Inhibitor, Cooperates with Ublituximab-Driven ADCC and ADCP in In Vitro and In Vivo Models of Ibrutinib-Resistant Mantle Cell Lymphomaet al., Ribeiro MTG-1701American Association for Cancer Research Annual Meeting (AACR)2020american-association-for-cancer-research-annual-meeting-aacroncologytg-1701
06/12/2020Long term Results of a Phase I/ Ib Study of Ibrutinib in Combination with Umbralisib in Patients with Relapsed/Refractory CLL or MCLDavids M, et al.umbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2020congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/12/2020Safety and Activity of the Once Daily Selective Bruton Tyrosine Kinase (BTK) Inhibitor TG-1701 in Patients with Chronic Lymphocytic Leukemia (CLL) and LymphomaCheah C, et al.TG-1701Congress of the European Hematology Association (EHA)2020congress-of-the-european-hematology-association-ehaoncologytg-1701
05/29/2020Effect of Adding Ublituximab to Ibrutinib on PFS, ORR, and MRD Negativity in Previously Treated High-Risk Chronic Lymphocytic Leukemia: Final Results of the GENUINE Phase III Studyet al., Sharman Jublituximab (TG-1101)American Society of Clinical Oncology Annual Meeting (ASCO)2020american-society-of-clinical-oncology-annual-meeting-ascooncologyublituximab-tg-1101
04/30/2020A Phase 2 Multicenter Study of Ublituximab, a Novel Glycoengineered Anti-CD20 Monoclonal Antibody, in Patients With Relapsing Forms of Multiple Sclerosiset al., Fox Eublituximab (TG-1101)Multiple Sclerosis Journal2020multiple-sclerosis-journalautoimmuneublituximab-tg-1101
02/27/2020Long-term Follow-up Results From the Phase 2 Multicenter Study of Ublituximab(UTX), a Novel Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), in Patients With Relapsing Multiple Sclerosis (RMS)et al., Fox Eublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2020americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
12/09/2019Phase 1 Study of TG-1701, a Selective Irreversible Inhibitor of Bruton’s Tyrosine Kinase (BTK), in Patients with Relapsed/Refractory B-Cell MalignanciesCheah C, et al.ublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2019american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/08/2019A Phase 1/2 Study of Umbralisib, Ublituximab and Venetoclax in Patients with Relapsed or Refractory Chronic Lymphocytic Leukemia (CLL).Barr P, et al.umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2019american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
11/21/2019Ublituximab and Umbralisib in Relapsed/Refractory B-cell Non-Hodgkin Lymphoma and Chronic Lymphocytic Leukemiaet al., Lunning Mumbralisib (TGR-1202)Blood Medical Journal – published by the American Society of Hematology (Blood)2019blood-medical-journal-published-by-the-american-society-of-hematology-bloodoncologyumbralisib-tgr-1202
09/23/2019A Phase 2 Study to Assess the Safety and Efficacy of Umbralisib in Patients with Chronic Lymphocytic Leukemia (CLL) Who Are Intolerant to Prior BTK or PI3K Delta Inhibitor Therapyet al., Mato Aumbralisib (TGR-1202)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2019international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyumbralisib-tgr-1202
09/23/2019Phase I/II Triple Therapy Study of Umbralisib and Ublituximab (U2) Combined with Checkpoint Inhibition in Patients with Relapsed/Refractory Chronic Lymphocytic Leukemia (CLL) and Richter’s Transformation (RT)et al., Mato Aumbralisib (TGR-1202)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2019international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyumbralisib-tgr-1202
09/12/2019Long-term Follow-up Results from the Phase 2 Multicenter Study of Ublituximab (UTX), a Novel Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), in Patients with Relapsing Multiple Sclerosis (RMS)et al., Fox Eublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2019european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
09/12/2019Study Design and Patient Demographics of the ULTIMATE Phase III Trials Evaluating Ublituximab (UTX), a Novel Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), in Patients with Relapsing Multiple Sclerosis (RMS)Cree B, et al.ublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2019european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
07/12/2019Open Label Extension (OLE) of Phase 2 Multicenter Study of Ublituximab (UTX), a Novel Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), in Patients with Relapsing Forms of Multiple Sclerosis (RMS)et al., Fox Eublituximab (TG-1101)5th Congress of the European Academy of Neurology (EAN)20195th-congress-of-the-european-academy-of-neurology-eanautoimmuneublituximab-tg-1101
06/20/2019Phase I/II Study of Umbralisib (TGR-1202) in Combination with Ublituximab (TG-1101) and Pembrolizumab in Patients with Relapsed/Refractory CLL and Richter’s Transformationet al., Mato Aublituximab (TG-1101), umbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2019international-congress-on-malignant-lymphoma-icmloncologyublituximab-tg-1101 umbralisib-tgr-1202
06/20/2019A Phase 2 Study to Assess the Safety and Efficacy of Umbralisib in Patients with Chronic Lymphocytic Leukemia (CLL) Who Are Intolerant to Prior BTK or PI3K Delta Inhibitor Therapyet al., Mato Aumbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2019international-congress-on-malignant-lymphoma-icmloncologyumbralisib-tgr-1202
06/19/2019Umbralisib Monotherapy Demonstrates Efficacy and Safety in Patients with Relapsed/Refractory Marginal Zone Lymphoma: A Multicenter, Open-Label, Registration Directed Phase 2 Studyet al., Zinzani Pumbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2019international-congress-on-malignant-lymphoma-icmloncologyumbralisib-tgr-1202
06/14/2019The Novel Bispecific CD47-CD19 Antibody TG-1801 Potentiates the Activity of Ublituximab-Umbralisib (U2) Drug Combination in Preclinical Models of B-NHLet al., Ribeiro MTG-1801Congress of the European Hematology Association (EHA)2019congress-of-the-european-hematology-association-ehaoncologytg-1801
06/09/2019The Novel Bispecific CD47-CD19 Antibody TG-1801 Potentiates the Activity of Ublituximab-Umbralisib (U2) Drug Combination in Preclinical Models of B-NHLet al., Ribeiro MTG-1801, ublituximab (TG-1101), umbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2019international-congress-on-malignant-lymphoma-icmloncologytg-1801 ublituximab-tg-1101 umbralisib-tgr-1202
06/04/2019Umbralisib Monotherapy Demonstrates Efficacy and Safety in Patients with Relapsed/Refractory Marginal Zone Lymphoma: A Multicenter, Open-label, Registration Directed Phase 2 Studyet al., Fowler Numbralisib (TGR-1202)American Society of Clinical Oncology Annual Meeting (ASCO)2019american-society-of-clinical-oncology-annual-meeting-ascooncologyumbralisib-tgr-1202
05/07/2019Open Label Extension (OLE) of a Phase 2 Multicenter Study Of Ublituximab, a Novel Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), in Patients with Relapsing Forms of Multiple Sclerosis (RMS)et al., Fox Eublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2019american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
05/03/2019B cell Depletion with Ublituximab Reshapes the T Cell Profile in Multiple Sclerosis Patientset al., Lovett-Racke Aublituximab (TG-1101)Journal of Neuroimmunology2019journal-of-neuroimmunologyautoimmuneublituximab-tg-1101
04/01/2019TG Therapeutics Reports Positive Interim Data from UNITY-NHL Phase 2b Trial Evaluating Umbralisib Monotherapy in Patients with Marginal Zone Lymphoma at the 2019 AACR Annual Meetinget al., Fowler Numbralisib (TGR-1202)American Association for Cancer Research Annual Meeting (AACR)2019american-association-for-cancer-research-annual-meeting-aacroncologyumbralisib-tgr-1202
02/28/2019Final Results of a Phase 2 Multicenter Study of Ublituximab, a Novel Glycoengineered Anti-CD20 Monoclonal Antibody, in Patients with Relapsing Forms of Multiple Sclerosis (RMS)et al., Fox Eublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2019americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
02/01/2019Tolerability and Activity of Ublituximab, Umbralisib, and Ibrutinib in Patients with Chronic Lymphocytic Leukaemia and Non-Hodgkin Lymphoma: A Phase 1 Dose Escalation and Expansion Trialet al., Nastoupil Lumbralisib (TGR-1202)New England Journal of Medicine (NEJM)2019new-england-journal-of-medicine-nejmoncologyumbralisib-tgr-1202
12/14/2018Umbralisib in Combination with Ibrutinib in Patients with Relapsed or Refractory Chronic Lymphocytic Leukaemia or Mantle Cell Lymphoma: A Multicentre Phase 1–1b StudyDavids M, et al.umbralisib (TGR-1202)THE LANCET Haematology2018the-lancet-haematologyoncologyumbralisib-tgr-1202
12/03/2018Combination of Umbralisib, Ublituximab, and Bendamustine is Safe and Highly Active in Patients with Advanced DLBCL and Follicular Lymphomaet al., Lunning Mublituximab (TG-1101), umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2018american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202
12/02/2018Phase I/II Study of Umbralisib (TGR-1202) in Combination with Ublituximab (TG-1101) and Pembrolizumab in Patients with Relapsed/Refractory CLL and Richter’s Transformationet al., Mato Aumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2018american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
10/11/2018Final Results of a Placebo Controlled, Phase 2 Multicenter Study of Ublituximab (UTX), a Novel Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), in Patients with Relapsing Forms of Multiple Sclerosis (RMS)et al., Fox Eublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2018european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
06/18/2018Phase 2 Multicenter Study Results of Ublituximab, a Novel Glycoengineered AntiCD20 Monoclonal Antibody (mAb), in Patients with Relapsing Multiple Sclerosis (RMS)et al., Fox Eublituximab (TG-1101)Congress of the European Academy of Neurology (EAN)2018congress-of-the-european-academy-of-neurology-eanautoimmuneublituximab-tg-1101
06/16/2018Resurrecting response to ruxolitinib: A Phase I study of ruxolitinib and umbralisib (TGR-1202) in ruxolitinib-experienced myelofibrosisMoyo et al.umbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2018congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/16/2018A Phase 2 Study to Assess the Safety and Efficacy of Umbralisib (TGR-1202) in Patients with Chronic Lymphocytic Leukemia (CLL) who are Intolerant to Prior BTK or PI3K Delta Inhibitor Therapyet al., Mato Aumbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2018congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/15/2018Long Term Integrated Safety Analysis Of Umbralisib (TGR-1202), A PI3K?/Ck1? Inhibitor With A Differentiated Safety Profile, In Patients With Relapsed/Refractory Lymphoid MalignanciesDavids M, et al.umbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2018congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/15/2018TG-1701 is a novel, orally available and covalently bound BTK inhibitorE et al., NormantTG-1701Congress of the European Hematology Association (EHA)2018congress-of-the-european-hematology-association-ehaoncologytg-1701
06/04/2018A Phase 2 Study to Assess the Safety and Efficacy of Umbralisib (TGR-1202) in Patients with CLL who are Intolerant to Prior BTK or PI3K Inhibitor Therapyet al., Mato Aumbralisib (TGR-1202)American Society of Clinical Oncology Annual Meeting (ASCO)2018american-society-of-clinical-oncology-annual-meeting-ascooncologyumbralisib-tgr-1202
04/24/2018Final MRI Results at 6 Months from a Phase 2 Multicenter Study of Ublituximab, A Novel Glyocoengineered Anti-CD20 Monoclonal Antibody (mAb), in Patients with Relapsing Forms of Multiple Sclerosis (RMS), Demonstrates Complete Elimination of Gd-Enhancing Lesionset al., Inglese Mublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2018american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/18/2018TG-1601 is a Novel BET Inhibitor with Strong Binding Affinity and Long-lasting Effect in Pre-clinical ModelsE et al., NormantTG-1601American Association for Cancer Research Annual Meeting (AACR)2018american-association-for-cancer-research-annual-meeting-aacroncologytg-1601
02/20/2018Umbralisib, a Novel PI3Kδ and Casein Kinase-1ε Inhibitor, in Relapsed or Refractory Chronic Lymphocytic Leukaemia and Lymphoma: an Open-label, Phase 1, Dose-escalation, First-in-human StudyBurris H, et al.umbralisib (TGR-1202)THE LANCET Oncology2018the-lancet-oncologyoncologyumbralisib-tgr-1202
02/01/20186 Month Results of a Phase 2a Multicenter Study of Ublituximab, a Novel Glycoengineered Anti-CD20 Monoclonal Antibody, in Relapsing Multiple Sclerosiset al., Fox Eublituximab (TG-1101)Americas Committee for Treatment and Research in Multiple Sclerosis (ACTRIMS)2018americas-committee-for-treatment-and-research-in-multiple-sclerosis-actrimsautoimmuneublituximab-tg-1101
12/11/2017KI Intolerance Study: A Phase 2 Study to Assess the Safety and Efficacy of Umbralisib (TGR-1202) in Patients with Chronic Lymphocytic Leukemia (CLL) Who Are Intolerant to Prior BTK or PI3K Delta Inhibitor Therapyet al., Mato Aumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2017american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/11/2017An Integrated Safety Analysis of the Next Generation PI3K Delta Inhibitor Umbralisib (TGR-1202) in Patients with Relapsed/Refractory Lymphoid MalignanciesDavids M, et al.umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2017american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/11/2017PI3K-Delta Inhibitors Induce Primary Monocyte Cytotoxicity but Do Not Alter Monocyte DifferentiationD et al, Friedmanumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2017american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/10/2017Phase I/II Study of Pembrolizumab in Combination with Ublituximab (TG-1101) and Umbralisib (TGR-1202) in Patients with Relapsed/Refractory CLLet al., Mato Aublituximab (TG-1101), umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2017american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101 umbralisib-tgr-1202
12/10/2017Umbralisib/TGR-1202 as a Novel Dual PI3K/CK1 Inhibitor Has a Unique Therapeutic Role in Silencing Oncogenes in Aggressive Lymphomaset al., O'Connorumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2017american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/10/2017Differential Regulation of T Cells By PI3K Delta Inhibitors in a CLL Murine Modelet al., Maharajumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2017american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
10/27/2017Placebo controlled, phase 2a multicenter study of ublituximab (UTX), a novel glycoengineered anti-CD20 monoclonal antibody (mAb), in patients with relapsing forms of multiple sclerosis (RMS): 6 months analysis of B cell subsetset al., Fox E, Lovett-Racke Aublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2017european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/26/2017Patient characteristics, safety, and preliminary results of a placebo controlled, phase 2a multicenter study of ublituximab (UTX), a novel glycoengineered anti-CD20 monoclonal antibody (mAb), in patients with relapsing forms of multiple sclerosiset al., Fox Eublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2017european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
10/26/2017Preliminary results of phase 2 multicenter study of ublituximab (UTX), a novel glycoengineered anti-CD20 monoclonal antibody (mAb), in patients with relapsing forms of multiple sclerosis (RMS) demonstrates rapid Gd-enhancing lesions decreaseet al., Inglese Mublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2017european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
06/24/2017Tolerability and activity of chemo-free triplet combination of umbralisib (TGR-1202), ublituximab, and ibrutinib in patients with advanced CLL and NHLet al., Nastoupil Lumbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2017congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/24/2017Combination of TGR-1202, Ublituximab, and bendamustine is safe and highly active in patients with advanced DLBCL and follicular lymphomaet al., Lunning Mublituximab (TG-1101)Congress of the European Hematology Association (EHA)2017congress-of-the-european-hematology-association-ehaoncologyublituximab-tg-1101
06/24/2017Rapid and Robust B Cell Depletion in Preliminary Results of Phase 2 Multicenter Study of Ublituximab (UTX), a Novel Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), in Patients with Relapsing forms of Multiple Sclerosis (RMS)et al., Fox Eublituximab (TG-1101)Congress of the European Academy of Neurology (EAN)2017congress-of-the-european-academy-of-neurology-eanautoimmuneublituximab-tg-1101
06/16/2017Ublituximab and ibrutinib for previously treated genetically high-risk chronic lymphocytic leukemia: Results of the GENUINE Phase 3 studyet al., Mato Aublituximab (TG-1101)International Congress on Malignant Lymphoma (ICML)2017international-congress-on-malignant-lymphoma-icmloncologyublituximab-tg-1101
06/16/2017Tolerability and activity of chemo-free triplet combination of umbralisib (TGR-1202), ublituximab, and ibrutinib in patients with advanced CLL and NHLet al., Nastoupil Lublituximab (TG-1101), umbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2017international-congress-on-malignant-lymphoma-icmloncologyublituximab-tg-1101 umbralisib-tgr-1202
06/15/2017Combination of TGR-1202, Ublituximab, and Bendamustine is safe and highly active in patients with advanced DLBCL and Follicular Lymphomaet al., Lunning Mumbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2017international-congress-on-malignant-lymphoma-icmloncologyumbralisib-tgr-1202
06/14/2017Updated Results of a Multicenter Phase I/IB Study of Umbralisib (TGR-1202) in Combination with Ibrutinib in Patients with Relapsed or Refractory MCL or CLLDavids M, et al.umbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2017international-congress-on-malignant-lymphoma-icmloncologyumbralisib-tgr-1202
06/05/2017Tolerability and activity of chemo-free triplet combination of TGR-1202, ublituximab, and ibrutinib in patients with advanced CLL and NHLet al., Nastoupil Lumbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2017congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/03/2017Ublituximab and ibrutinib for previously treated genetically high-risk chronic lymphocytic leukemia: Results of the GENUINE Phase 3 studyet al., Sharman Jublituximab (TG-1101)American Society of Clinical Oncology Annual Meeting (ASCO)2017american-society-of-clinical-oncology-annual-meeting-ascooncologyublituximab-tg-1101
05/26/2017Rapid and Robust B Cell Depletion in Preliminary Results of a Phase 2 Study of Ublituximab, Novel Glycoengineered Anti-CD20 Mab, RMS Patientset al., Fox E, Lovett-Racke Aublituximab (TG-1101)Annual Meeting of Consortium of MS Centers (CMSC)2017annual-meeting-of-consortium-of-ms-centers-cmscautoimmuneublituximab-tg-1101
05/15/2017TGR-1202– A novel PI3K-delta inhibitor that differentially regulates T cells in CLLet al., Pinilla-Ibarzumbralisib (TGR-1202)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2017international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyumbralisib-tgr-1202
05/15/2017TGR-1202 in Combination with Ibrutinib in Patients with Relapsed or Refractory CLL: Updated Results of a Multicenter Phase I/Ib StudyDavids M, et al.umbralisib (TGR-1202)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2017international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyumbralisib-tgr-1202
04/28/2017Preliminary results of Phase 2 Multicenter Study of Ublituximab (UTX), a novel glycoengineered anti-CD20 monoclonal antibody (mAb), in patients with relapsing forms of Multiple Sclerosis (RMS) demonstrates rapid and robust B cell depletionet al., Fox E, Lovett-Racke Aublituximab (TG-1101)American Academy of Neurology Annual Meeting (AAN)2017american-academy-of-neurology-annual-meeting-aanautoimmuneublituximab-tg-1101
04/04/2017Preclinical Characterization of a Fully Human lgG1 Anti PD-L1 mab CK-301et al., Gorelik L, Marasco WAnti PD-L1American Association for Cancer Research Annual Meeting (AACR)2017american-association-for-cancer-research-annual-meeting-aacroncologyanti-pd-l1
03/05/2017KI intolerance study: A phase 2 study to assess the safety and efficacy of TGR-1202 in pts with chronic lymphocytic leukemia (CLL) who are intolerant to prior BTK or PI3K-delta inhibitor therapyDorsey, et al., Matoumbralisib (TGR-1202)American Society of Clinical Oncology Annual Meeting (ASCO)2017american-society-of-clinical-oncology-annual-meeting-ascooncologyumbralisib-tgr-1202
02/21/2017Ublituximab (TG-1101), a novel glycoengineered anti-CD20 antibody, in combination with ibrutinib is safe and highly active in patients with relapsed and/or refractory chronic lymphocytic leukaemia: results of a phase 2 trialBurke et al., Sharmanublituximab (TG-1101)British Journal of Haematology (BJH)2017british-journal-of-haematology-bjhoncologyublituximab-tg-1101
12/16/2016A phase 1/2 trial of ublituximab, a novel, glycoengineered anti-CD20 monoclonal antibody, in patients with B-cell non-Hodgkin lymphoma or chronic lymphocytic leukaemia previously exposed to rituximabet al., O'Connor, Sawasublituximab (TG-1101)British Journal of Haematology (BJH)2016british-journal-of-haematology-bjhoncologyublituximab-tg-1101
12/05/2016TGR-1202 in Combination with Ibrutinib in Patients with Relapsed or Refractory CLL or MCL: Preliminary Results of a Multicenter Phase I/Ib Study.Davids M, et al.umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2016american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/05/2016Preliminary Results from a Phase I Dose Escalation Trial of Ruxolitinib and the PI3K Delta Inhibitor TGR-1202 in Myelofibrosis.Moyo et al.umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2016american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/05/2016Combination of Ublituximab, TGR-1202 and Bendamustine Demonstrates Significant Activity in Patients with Advanced DLBCL and Follicular Lymphoma.et al., Lunning Mumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2016american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/05/2016A Phase I Trial of TGR-1202, a Next Generation Once Daily PI3K Delta Inhibitor, in Combination with Brentuximab Vedotin, in Patients with Relapsed/Refractory Hodgkins LymphomaRamchandran et al.umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2016american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/04/2016Silencing cMyc Translation as a Therapeutic Strategy Through Targeting PI3K Delta and CK1 Epsilon in Hematological Malignancies.Deng C, et al.umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2016american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/04/2016Modulation of T cell Compartment in a Preclinical CLL Murine Model by a Selective PI3K delta inhibitor, TGR-1202.et al., Maharajumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2016american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
10/27/2016Silencing c-Myc Translation as a Therapeutic Strategy through Targeting PI3K Delta and CK1 Epsilon in Hematological MalignanciesDeng C, et al., O'Connor Oumbralisib (TGR-1202)Blood Medical Journal – published by the American Society of Hematology (Blood)2016blood-medical-journal-published-by-the-american-society-of-hematology-bloodoncologyumbralisib-tgr-1202
09/14/2016Open Label Safety Study of Ublituximab for the Treatment of Acute Neuromyelitis Optica Relapseset al., Levy M, Mealy Mublituximab (TG-1101)European Committee for Treatment and Research in Multiple Sclerosis (ECTRIMS)2016european-committee-for-treatment-and-research-in-multiple-sclerosis-ectrimsautoimmuneublituximab-tg-1101
06/03/2016Long-term follow-up of the PI3K delta inhibitor TGR-1202 demonstrates a differentiated safety profile and high response rates in CLL and NHL: Integrated-analysis of TGR-1202 monotherapy and combined with ublituximab.Burris H, et al., Flinn Iumbralisib (TGR-1202)American Society of Clinical Oncology Annual Meeting (ASCO)2016american-society-of-clinical-oncology-annual-meeting-ascooncologyumbralisib-tgr-1202
06/01/2016Preliminary Results of a Phase I/Ib Study of Ibrutinib in Combination with TGR-1202 in Patients with Relapsed/Refractory CLL or MCL.Davids M, et al.umbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2016congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/01/2016Long-term follow-up of the PI3k delta inhibitor TGR-1202 demonstrates a differentiated safety profile and high response rates in CLL: Integrated-analysis of TGR-1202 monotherapy and combined with ublituximab.et al., Mato Aumbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2016congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/01/2016Long-term follow-up of PI3K delta inhibitor TGR-1202 demonstrates safety and high response rates in NHL: Integrated Analysis of TGR-1202 monotherapy and combined with ublituximabet al., O'Connor Oumbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2016congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
04/16/2016Differential Regulation of Human T cells by TGR-1202, A Novel PI3K-delta Inhibitor.et al., Pinilla-Ibarzumbralisib (TGR-1202)American Association for Cancer Research Annual Meeting (AACR)2016american-association-for-cancer-research-annual-meeting-aacroncologyumbralisib-tgr-1202
12/08/2015Ublituximab (TG-1101), a Novel Glycoengineered Anti-CD20 Monoclonal Antibody, in Combination with Ibrutinib is Highly Active in Patients with Relapsed and/or Refractory Mantle Cell Lymphoma: Results of a Phase II Trial.et al., Sharman Jublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2015american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/08/2015Disruption of the mTOR-eIF4F Axis By Selectively Targeting PI3Kdelta and Proteasome Potently Inhibits Cap Dependent Translation of c-Myc in Aggressive Lymphomas.Deng C, et al.umbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2015american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/08/2015Clinical Activity and Safety Profile of TGR-1202, a Novel Once Daily PI3K- Delta Inhibitor, in Patients with CLL and B-Cell Lymphoma.et al., O'Connor Oumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2015american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/08/2015A Phase I Trial of TGR-1202, a Next Generation Once Daily PI3K-Delta Inhibitor in Combination with Obinutuzumab Plus Chlorambucil, in Patients with Chronic Lymphocytic Leukemia.et al., Mahadevan Dumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/08/2015A Phase I Trial of TGR-1202, a Next Generation Once Daily PI3K-Delta Inhibitor in Combination with Obinutuzumab Plus Chlorambucil, in Patients with Chronic Lymphocytic Leukemia.et al., Mahadevan Dumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2015american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
11/08/2015Ublituximab (TG-1101), a Novel Glycoengineered Anti-CD20 Monoclonal Antibody, in Combination with Ibrutinib is Highly Active in Patients with Relapsed and/or Refractory Mantle Cell Lymphoma: Results of a Phase II Trial.et al., Sharman Jublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2015american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
09/09/2015a Novel Once Daily PI3K-Delta Inhibitor, Demonstrates Clinical Activity with a Favorable& Differentiated Safety Profile as a Single Agent and in Combination with a Novel Glyocengineered anti-CD20 mAb, Ublituximab in Patients with Rel/Ref CLL.et al., O'Brienublituximab (TG-1101)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyublituximab-tg-1101
09/09/2015a Novel Once Daily PI3K-Delta Inhibitor, Demonstrates Clinical Activity with a Favorable& Differentiated Safety Profile as a Single Agent and in Combination with a Novel Glyocengineered anti-CD20 mAb, Ublituximab in Patients with Rel/Ref CLL.et al., O'Brienublituximab (TG-1101)International Workshop on Chronic Lymphocytic Leukemia (iwCLL)2015international-workshop-on-chronic-lymphocytic-leukemia-iwclloncologyublituximab-tg-1101
06/20/2015Ublituximab + TGR-1202 Demonstrates Activity and Favorable Safety Profile in Relapsed/Refractory B-Cell NHL and High-Risk CLL.et al., Lunning Mumbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2015international-congress-on-malignant-lymphoma-icmloncologyumbralisib-tgr-1202
06/20/2015Ublituximab (TG-1101), a Novel Glycoengineered Anti-CD20 MAB, in Combination with Ibrutinib Achieves 95% ORR in Patients with High-Risk Relapsed/Refractory CLL.Burke J, et al.ublituximab (TG-1101)International Congress on Malignant Lymphoma (ICML)2015international-congress-on-malignant-lymphoma-icmloncologyublituximab-tg-1101
06/20/2015Safety and Activity of the Chemotherapy-Free Triplet of Ublituximab, TGR-1202, and Ibrutinib is Safe and Highly Active in Relapsed B-Cell Malignancies.et al., Nastoupil Lumbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2015international-congress-on-malignant-lymphoma-icmloncologyumbralisib-tgr-1202
06/20/2015Clinical Activity and Safety Profile of TGR-1202, a Novel Once Daily PI3K-Delta Inhibitor, Demonstrates Clinical Activity with a Favorable Safety Profile, Lacking Hepatotoxicity in Patients with CLL and B-Cell Lymphoma.et al., O'Connorumbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2015international-congress-on-malignant-lymphoma-icmloncologyumbralisib-tgr-1202
06/14/2015Ublituximab + TGR-1202 Demonstrates Activity and Favorable Safety Profile in Relapsed/Refractory B-Cell NHL and High-Risk CLL.et al., Lunning Mublituximab (TG-1101)Congress of the European Hematology Association (EHA)2015congress-of-the-european-hematology-association-ehaoncologyublituximab-tg-1101
06/14/2015Clinical Activity and Safety Profile of TGR-1202 a Novel Once Daily PI3K-Delta Inhibitor, Demonstrates Clinical Activity with a Favorable Safety Profile, Lacking Hepatotoxicity, in Patients with CLL and B-Cell Lymphoma.et al., O'Connorumbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2015congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/02/2015Ubliuximab +TGR-1202 Demonstrates Activity and Favorable Safety Profile in Relapsed/Refractory B-Cell NHL and High-Risk CLL.et al., Lunning M, O'Brien Sumbralisib (TGR-1202)American Society of Clinical Oncology Annual Meeting (ASCO)2015american-society-of-clinical-oncology-annual-meeting-ascooncologyumbralisib-tgr-1202
06/02/2015Safety and Activity of the Chemotherapy-free Triplet of Ublituximab, TGR-1202 and ibrutinib in Relapsed B-cell Malignancies.et al., Fowler N, O'Brien Sublituximab (TG-1101)American Society of Clinical Oncology Annual Meeting (ASCO)2015american-society-of-clinical-oncology-annual-meeting-ascooncologyublituximab-tg-1101
06/02/2015Clinical Activity and Safety Profile of TGR-1202, a Novel Once Daily Pi3k Delta Inhibitor, in Patients with CLL and B-Cell Lymphoma.Burris H, et al., Flinn Iumbralisib (TGR-1202)American Society of Clinical Oncology Annual Meeting (ASCO)2015american-society-of-clinical-oncology-annual-meeting-ascooncologyumbralisib-tgr-1202
04/18/2015IRAK4 inhibitors display synergistic activity when combined with BTK or PI3K inhibitors in B-cell lymphomas.et al., Marschke K, Vajda EIRAK4American Association for Cancer Research Annual Meeting (AACR)2015american-association-for-cancer-research-annual-meeting-aacroncologyirak4
03/08/2015Ublituximab + TGR-1202 Demonstrates Activity and a Favorable Safety Profile in Relapsed/Refractory B-Cell NHL and High-Risk CLL: Phase I Results.et al., Lunning Mumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2015american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/09/2014Ublituximab, a Novel Glycoengineered Anti-CD20 Monoclonal Antibody (mAb), in Combination with TGR-1202, a Next Generation Once Daily PI3K Delta Inhibitor, Demonstrate Activity in Heavily Pre-Treated and High-Risk Chronic Lymphocytic Leukemia (CLL) and B-Cell Lymphoma.et al., Lunning M, O'Brien Sumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2014american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/09/2014Ublituximab (TG-1101) a Novel Glycoengineered Anti-CD20 Monoclonal Antibody, in Combination with Ibrutinib is Highly Active in Patients with Relapsed and/or Refractory CLL and MCL: Results of a Phase II Trial.et al., Greenwald D, Sharman Jublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2014american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/09/2014The PI3K-delta Inhibitor TGR-1202 in Combination with Brentuximab Vedotin (SGN-35) Synergistically Inhibits Tubulin Polymerization and Exerts Potent Antitumor Effects in NOD/SCID Mice with Hodgkin Lymphoma Cell Line Xenografts.et al., Locatelliumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2014american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/09/2014TGR-1202, a Novel Once Daily Pi3K Delta Inhibitor, Demonstrates Clinical Activity with a Favorable Safety Profile, Lacking Hepatotoxicity, in Patients with Chronic Lymphocytic Leukemia and B-Cell Lymphoma.Burris H, et al., Flinn Iumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2014american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/09/2014Complementary Targeting of PI3K and the Proteasome Causes Potent Inhibition of mTORC1 and NF-kappaB in Models of B- and T-Cell Lymphoma.Deng C, et al., O'Connor Oumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2014american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
07/21/2014A Phase I Trial of Ublituximab, A Novel Glycoengineered Anti-CD20 mAb, In Combination With TGR-1202, A Next Generation PI3K Delta Inhibitor, In Patients With Chronic Lymphocytic Leukemia And Non-Hodgkin’s Lymphoma.et al., Lunning M, O'Brien Sublituximab (TG-1101)Pan Pacific Lymphoma Conference (PPLC)2014pan-pacific-lymphoma-conference-pplconcologyublituximab-tg-1101
06/13/2014Ublituximab (TG-1101), A Novel Glycoenginereed Anti-CD20 mAb, in Combination with Ibrutinib in Patients with CLL and MCL; Results of an Ongoing Phase II Trial.et al., O'Connor O, Sharman Jublituximab (TG-1101)Congress of the European Hematology Association (EHA)2014congress-of-the-european-hematology-association-ehaoncologyublituximab-tg-1101
06/13/2014Ublituximab (TG-1101), A Novel Anti-CD20 Monoclonal Antibody for Rituximab Relapsed/Refractory B-Cell Malignancies.et al., Farber C, O'Connor Oublituximab (TG-1101)Congress of the European Hematology Association (EHA)2014congress-of-the-european-hematology-association-ehaoncologyublituximab-tg-1101
06/13/2014Activity of TGR-1202, a Novel Once-Daily Pi3K Delta Inhibitor, in Patients with Relapsed or Refractory Hematologic Malignancies.Burris H, et al., Flinn Iumbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2014congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
05/30/2014Activity of TGR-1202, a Novel Once-Daily Pi3K Delta Inhibitor, in Patients with Relapsed or Refractory Hematologic Malignancies.Burris H, et al., Flinn Iumbralisib (TGR-1202)American Society of Clinical Oncology Annual Meeting (ASCO)2014american-society-of-clinical-oncology-annual-meeting-ascooncologyumbralisib-tgr-1202
05/30/2014A Phase I Trial of Ublituximab (TG-1101), a Novel Anti-CD20 Monoclonal Antibody (MAB) in B-Cell Lymphoma Patients with Prior Exposure to Rituximab.Changchun D, et al., O'Connor Oublituximab (TG-1101)American Society of Clinical Oncology Annual Meeting (ASCO)2014american-society-of-clinical-oncology-annual-meeting-ascooncologyublituximab-tg-1101
04/09/2014The PI3K Delta Inhibitor TGR-1202 Induces Cytotoxicity and Inhibits Phosphorylation of AKT in 17p Deleted and Non-17p Deleted CLL Cells in Vitro.et al., Friedman D, Lanasa Mumbralisib (TGR-1202)American Association for Cancer Research Annual Meeting (AACR)2014american-association-for-cancer-research-annual-meeting-aacroncologyumbralisib-tgr-1202
04/09/2014The PI3K Delta Inhibitor TGR-1202 In Combination with Brentuximab Vedotin (SGN-35) Synergistically Induces G2/M Phase Arrest and Cell Death Via Inhibition of Tubulin Polymerization in Hodgkin Lymphoma Cell Lines.Carlo-Stella C, et al., Locatelli Sumbralisib (TGR-1202)American Association for Cancer Research Annual Meeting (AACR)2014american-association-for-cancer-research-annual-meeting-aacroncologyumbralisib-tgr-1202
12/10/2013The PI3K-d Inhibitor TGR-1202 in Combination with Brentuximab Vedotin (SGN-35) Synergistically Induces G2/M Phase Arrest and Cell Death Via Inhibition Of Tubulin Polymerization in Hodgkin Lymphoma Cell Lines.Carlo-Stella C, et al., Locatelli Sumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2013american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/10/2013The PI3K Delta Inhibitor TGR-1202 and Proteasome Inhibitor Carfilzomib are Highly Synergistic in Killing Human B- and T-Cell Lymphoma Cells.Deng C, et al., O'Connor Oumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2013american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/10/2013A Phase I Dose Escalation Study of TGR-1202, a Novel PI3K-d Inhibitor, For Patients with Relapsed or Refractory Hematologic Malignancies.et al., Patel M, Savona Mumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2013american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
09/09/2013The PI3k-delta inhibitor TGR-1202 induces cytotoxicity and inhibits phosphorylation of AKT in 17p deleted and non-17p deleted CLL cells in vitro.et al., Friedman D, Lanasa Mumbralisib (TGR-1202)American Association for Cancer Research Annual Meeting (AACR)2013american-association-for-cancer-research-annual-meeting-aacroncologyumbralisib-tgr-1202
06/14/2013Ublituximab (TG-1101), a Novel Anti-CD20 Monoclonal for Rituximab Relapsed/Refractory B-cell Malignancies.Changchun D, et al., O'Connor Oublituximab (TG-1101)Congress of the European Hematology Association (EHA)2013congress-of-the-european-hematology-association-ehaoncologyublituximab-tg-1101
06/14/2013A Novel, PI3K-Delta Specific Inhibitor in Multiple Myeloma.et al., Vakkalanka S, Viswanadha Sumbralisib (TGR-1202)Congress of the European Hematology Association (EHA)2013congress-of-the-european-hematology-association-ehaoncologyumbralisib-tgr-1202
06/04/2013Final Results of a Multicenter Phase Ib Single Agent Study with the Novel Anti-CD20 Monoclonal Antibody Ublituximab (TG-1101) in Patients with Relapsed Chronic Lymphocytic Leukemia (CLL).Cazin B, et al., Ribrag Vublituximab (TG-1101)Congress of the European Hematology Association (EHA)2013congress-of-the-european-hematology-association-ehaoncologyublituximab-tg-1101
06/02/2013A Phase I Dose-Escalation Trial of Ublituximab (TG-1101), a Novel Anti-CD20 Monoclonal Antibody (mAb) for Rituximab Relapsed and/or Refractory C-Cell Lymphoma Patients.Changchun D, et al., O'Connor Oublituximab (TG-1101)American Society of Clinical Oncology Annual Meeting (ASCO)2013american-society-of-clinical-oncology-annual-meeting-ascooncologyublituximab-tg-1101
06/01/2013Novel PI3K Inhibitors Demonstrate Marked Cytotoxicity in Models of T-Cell Lymphoma, Caused Apoptosis and Were Synergistic with the Novel Anti-CD20 Monoclonal Antibody Ublituximab in Models of B-Cell LymphomaChangchun, Dengumbralisib (TGR-1202)International Congress on Malignant Lymphoma (ICML)2013international-congress-on-malignant-lymphoma-icmloncologyumbralisib-tgr-1202
03/10/2013Combined Carfilzomib and Selective PI3K-d Inhibition (TGR-1202) Results in Enhanced Myeloma Cell Apoptosis.et al., Lonial S, Torre Cumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2013american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/11/2012Ublituximab, an Optimized Anti-CD20 Monoclonal Antibody, Demonstrates Greater NK-Mediated ADCC Than Rituximab in Waldenstrom’s Macroglobulinemia Patients Supporting a Therapeutic Strategy with Ublituximab.et al., Le Garff-Tavernier M, Leblond Vublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2012american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/11/2012Ublituximab (TGTX-1101), a Novel, Third-Generation Anti-CD20 Antibody Demonstrates Enhanced Antitumor Activity Compared to Rituximab in Primary CNS and Intraocular Lymphoma Murine Models.Donnou S, et al., Fisson Sublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2012american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/11/2012Ublituximab (TGTX-1101), A Novel Anti-CD20 Monoclonal Antibody (mAb), Demonstrates Activity in Rituximab-sensitive and Rituximab–resistant B Non-Hodgkin Lymphoma (B-NHL) Pre-clinical In Vitro and In Vivo Models.Barth M, Czuczman M, et al.ublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2012american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/11/2012TGR-1202 Suppresses AML and ALL Cells Via Selective Inhibition of PI3K-delta Kinase.et al., Savona M, Vakkalanka Sumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2012american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/11/2012Novel PI3K Inhibitors Demonstrate Marked Cytotoxicity in Models of T-Cell Lymphoma, Caused Apoptosis and Were Synergistic with the Novel Anti-CD20 Monoclonal Antibody Ublituximab in Models of B-Cell LymphomaChangchun D, et al., O'Connor Oumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2012american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
12/11/2012Comparison of the PI3K-delta Inhibitors TGR1202 and GS-1101 in Inducing Cytotoxicity and Inhibiting Phosphorylation of Akt in CLL Cells in Vitro.et al., Friedman D, Lanasa M, Weinberg Bumbralisib (TGR-1202)American Society of Hematology Annual Meeting (ASH)2012american-society-of-hematology-annual-meeting-ashoncologyumbralisib-tgr-1202
04/04/2012Inhibition of PI3Kd kinase by a selective small molecule inhibitor suppresses B-cell proliferation and leukemic cell growth.et al., Vakkalanka S, Viswanadha Sumbralisib (TGR-1202)American Association for Cancer Research Annual Meeting (AACR)2012american-association-for-cancer-research-annual-meeting-aacroncologyumbralisib-tgr-1202
12/13/2011TG20, a Transgenically-Derived Anti-CD20 Monoclonal Antibody, Exhibits Enhanced Cytotoxicity Against Cells with Low Levels of CD20.Echelard Y, et al., Meade HMublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2011american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/13/2011Multicentre Phase I Study with an 8-Dose Regimen of Single Agent Anti-CD20 Monoclonal Antibody LFB-R603 in Patients with Relapsed Chronic Lymphocytic Leukemia (CLL).Cartron G, Cazin B, Coiffier B, et al.ublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2011american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/13/2011LFB-R603, a Third-Generation Monoclonal Anti-CD20 Antibody, Displays Additive Antitumor Activity with Antileukemic Chemotherapeutic Agents in Mouse Xenograft Models.et al., Fournès B, Tourais Esteves Iublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2011american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/13/2011Comparison of Cell Lysis Mediated by LFB-R603 with That Mediated by Ofatumumab Against Cells Expressing Low Levels of CD20.Bellon A, et al., Salcedo Mublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2011american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
12/07/2010A Phase I study of LFB-R603, a Novel Anti-CD20 Antibody, in Patients with Relapsed Chronic Lymphocytic Leukemia.Cartron G, Cazin B, et al.ublituximab (TG-1101)American Society of Hematology Annual Meeting (ASH)2010american-society-of-hematology-annual-meeting-ashoncologyublituximab-tg-1101
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